All publications

Size characterization of lipid-based self-emulsifying pharmaceutical excipients during lipolysis using Taylor dispersion analysis with fluorescence detection

  • Scientific publication

International Journal of Pharmaceutics, Volume 537, Issues 1–2, Pages 94–101 - Feb 2018

Joseph Chamieh, Habib Merdassi, Jean-Christophe Rossi, Vincent Jannin, Frédéric Demarne, Hervé Cottet

In this work, the lipolysis of Labrasol® and Gelucire® 44/14 , two lipid based self-emulsifying drug delivery systems, by pancreatic enzymes and under conditions mimicking the gastrointestinal tract is followed by Taylor dispersion analysis. Results show that, Labrasol® droplets decrease exponentially in size with lipolysis time, whereas Gelucire® 44/14 droplets increased sigmoïdally in size. Even after 120 min lipolysis, both systems maintain a solubilizing capacity of the hydrophobic marker.

Hydrodynamic size characterization of a self-emulsifying lipid pharmaceutical excipient by Taylor dispersion analysis with fluorescent detection

  • Scientific publication

International Journal of Pharmaceutics, Volume 513, Issues 1–2, Pages 262-269 - Nov 2016

Vincent Jannin, Frédéric Demarne, Hervé Cottet

In this study the size of microemulsion droplets is carried out using Tailor Dispersion Analysis in comparison to Dynamic Light Scattering. The size evolution of a Labrasol® self emulsifying drug delivery system as a function of concentration and temperature is evaluated. The influence of physical parameters and polydispersity is discussed.

In Vitro Digestion of the Self-Emulsifying Lipid Excipient Labrasol® by Gastrointestinal Lipases and Influence of its Colloidal Structure on Lipolysis Rate

  • Scientific publication

Pharmaceutical Research volume 30, pages 3077–3087 DOI: 10.1007/s11095-013-1053-0 - May 2013

Sylvie Fernande, Vincent Jannin, Stéphanie Chevrier, Yann Chavant, Frédéric Demarne, Frédéric Carrière

In vitro lipolysis of the self-emulsifying excipient, Labrasol®

  • Poster

AAPS Annual Meeting & Exposition – San Diego (USA)  - Nov 2007

Sylvie FERNANDEZ, Nicolas RITTER, Stéphanie CHEVRIER, Frédéric CARRIÈRE and Vincent JANNIN